Bazedoxifene-d4

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Catalog No.: PC0131

Size: 1 mg, 5 mg

Description

Bazedoxifene-d4 is deuterium-labeled Bazedoxifene, an oral, BBB-penetrating non-steroidal selective estrogen receptor modulator (SERM). Bazedoxifene is used in osteoporosis research. Bazedoxifene also serves as an inhibitor of the IL-6/GP130 protein-protein interaction and may be useful in pancreatic cancer research.

Molecular Weight	474.63
Formula	C30H30D4N2O3
CAS No.	1133695-49-4
SMILES	CC1=C(N(C2=C1C=C(C=C2)O)CC3=CC=C(C=C3)OC([2H])(C([2H])(N4CCCCCC4)[2H])[2H])C5=CC=C(C=C5)O
Shipping	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
*In Vitro*	Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

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